LD50 (Lethal Dose, 50%) refers to the dose of a substance required to kill 50% of a tested population under controlled conditions. It is typically expressed in milligrams of the substance per kilogram of body weight (mg/kg) for the subject being tested, such as animals in laboratory studies.
Key Points:
1. Purpose: LD50 is used to measure and compare the acute toxicity of different substances.
2. Testing Population: The test is usually conducted on a specific group of animals, such as mice or rats, but extrapolation to humans must be done cautiously.
3. Route of Administration: The LD50 value depends on the route of exposure (e.g., oral, inhalation, dermal) because different routes may affect absorption and toxicity.
4. Units: LD50 is often reported in mg/kg, meaning the amount of substance (in milligrams) required per kilogram of the test subject’s body weight to reach the lethal 50% threshold.
Example:
• If the oral LD50 of a substance is 300 mg/kg, a dose of 300 mg would theoretically be lethal for 50% of a population of 1 kg animals.
LD50 values are a benchmark in toxicology for comparing substances’ toxic potency, though ethical considerations have reduced its use in favor of alternative testing methods.
Aspirin
LD50 200 mg/kg (rat, oral)
Gastric distress, confusion, psychosis, stupor, ringing in ears, drowsiness, hyperventilation
Sodium chloride (Salt)
12357 mg/kg (human, oral)
Eye irritant, elevated blood pressure
Glucose (sugar)
LD50 30 g/kg (rat, oral)
Depressed activity, gastrointestinal disturbances. If diabetic- heart disease, blindness, nerve damage, kidney damage
Ethanol (alchohol)
LD50 7060 mg/kg (rat, oral)
Nausea, headache, vomiting, dizziness, nervous system depression, confusion, loss of consciousness
Caffeine
LD50 140 mg/kg (dog, oral)
Acute renal failure, nausea, psychosis, hemorrhage, increased pulse, convulsions